Synthesis of 4-aminotetrahydropyran scaffolds for drug discovery

The European Lead Factory: A Blueprint for Public–Private Partnerships in Early Drug Discovery

A. Karawajczyk, K.M. Orrling, J.B.S. de Vlieger, T. Rijnders and D. Tzalis
Front. Med. 2017 3 (75)
doi: 10.3389/fmed.2016.00075 2017 January 19

De Novo Assembly of Highly Substituted Morpholines and Piperazines

P. Patil, R. Madhavachary, K. Kurpiewska, J. Kalinowska-Tłuścik and A. Dömling
Org Lett
doi: 10.1021/acs.orglett.6b03807 2017 January 19

Synthesis of Epibatidine Analogues by Pyrrole Diels–Alder Reactions: Rapid Access to Azabicyclo[2.2.1]heptane and 3,8-Diazabicyclo[3.2.1]octane Scaffolds for Library Synthesis

A.T. Murray, E. Packard, A. Nortcliffe, W. Lewis, D. Hamza, G. Jones, C.J. Moody
Eur. J. Org. Chem. 2017, 138–148
doi: 10.1002/ejoc.201601177 2016 December 19

Discovery of novel inhibitors to investigate diacylglycerol lipases and α/β hydrolase domain 16A

Unconventional Passerini Reaction toward α‑Aminoxy-amides

Charting Biologically Relevant Spirocyclic Compound Space

G. Müller, T. Berkenbosch, J. Benningshof, D. Stumpfe, J. Bajorath
doi: 10.1002/chem.201604714 2016 November 8 (epub ahead of print)

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