Publications

This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication. 

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28 December 2015

Rapid and Scalable Access into Strained Scaffolds through Continuous Flow Photochemistry

Blanco-Ania D, Gawade SA, Zwinkels LJL, Maartense L, Bolster MG, Benningshof JCJ, and Rutjes FPJT
Org Process Res Dev, 2016, 20(2):409–413
doi: 10.1021/acs.oprd.5b00354 Epub 2015, Dec 28

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05 November 2015

The ELF Honest Data Broker: informatics enabling public–private collaboration in a precompetitive arena

G. Paillard, P. Cochrane, P. S. Jones, A. Caracoti, H. van Vlijmen, A. D. Pannifer
Drug Discovery Today 21 (1), 97–102
doi:10.1016/j.drudis.2015.11.005

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30 September 2015

Expansion of chemical space for collaborative lead generation and drug discovery – the European Lead Factory Perspective

A. Karawajczyk, F. Giordanetto, J. Benningshof, D. Hamza, T. Kalliokoski, K. Pouwer, R. Morgentin, A. Nelson, G. Müller, A. Piechot, D. Tzalis
Drug Discovery Today 20 (11), 1310–1316
doi: 10.1016/j.drudis.2015.09.009 Epub 2015 Sep 30

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30 September 2015

The importance of triaging in determining the quality of output from high-throughput screening

Jones PS, McElroy S,  Morrison A and Pannifer A.
Future Medicinal Chemistry 2015;7(14):1847-52. 
doi: 10.4155/fmc.15.121 Epub 2015 Sep 30

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26 September 2015

The European Lead Factory

Christopher Kallus, Jörg Hüser, Philip S. Jones, Adam Nelson
Chapter 2 in the book Small Molecule Medicinal Chemistry: Strategies and Technologies (ed. W. Czechtizky and P. Hamley) Wiley 
doi: https://doi.org/10.1002/9781118771723.ch2 2015 September 26

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15 September 2015

Price-focused Analysis of Commercially Available Building Blocks for Combinatorial Library Synthesis

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10 August 2015

Leuckart-Wallach Route Toward Isocyanides and Some Applications

C.G. Neochoritis, T. Zarganes-Tzitzikas, S. Stotani,A. Dömling, E. Herdtweck, K. Khoury and A. Dömling
ACS Comb. Sci.
doi: 10.1021/acscombsci.5b00066 Epub 2015, Aug 10

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03 August 2015

Leuckart-Wallach Approach to Sugar Isocyanides and Its IMCRs

C.G. Neochoritis, J. Zhang and A. Dömling
Synthesis 2015; 47(16): 2407-2413
doi: 10.1055/s-0034-1381046 Epub 2015 Aug 3

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30 July 2015

Synthesis of (Arylamido)pyrrolidinone Libraries through Ritter-Type Cascade Reactions of Dihydroxylactams

Wu P et al.
European Journal of Organic Chemistry, 2015 (25), 5633–5639 
doi: 10.1002/ejoc.201500712 ePub 2015 Jul 30

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09 July 2015

Facile Access to a Heterocyclic, sp3-Rich Chemical Scaffold via a Tandem Condensation/ Intramolecular Nitrone-Alkene [3+2] Cycloaddition Strategy

M. J. Rawling, T. E. Storr, W. A. Bawazir, S. J. Cully, W. Lewis, M. S. I. T. Makki,  I. R. Strutt, G. Jones, D. Hamza and R. A. Stockman
Chem. Commun., 2015, 51, 12867-12870
doi: 10.1039/C5CC05070G Epub 2015 Jul 9

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