Publications

This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication. 
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19 December 2016

Synthesis of Epibatidine Analogues by Pyrrole Diels–Alder Reactions: Rapid Access to Azabicyclo[2.2.1]heptane and 3,8-Diazabicyclo[3.2.1]octane Scaffolds for Library Synthesis

A.T. Murray, E. Packard, A. Nortcliffe, W. Lewis, D. Hamza, G. Jones, C.J. Moody
Eur. J. Org. Chem. 2017, 138–148
doi: 10.1002/ejoc.201601177 2016 December 19

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01 December 2016

Unconventional Passerini Reaction toward α‑Aminoxy-amides

A.L. Chandgude and A.S.S. Dömling
Org. Lett., 2016, 18 (24), pp 6396–6399
doi: 10.1021/acs.orglett.6b03293 2016 December 1

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01 December 2016

Discovery of novel inhibitors to investigate diacylglycerol lipases and α/β hydrolase domain 16A

F.J. Janssen
Doctoral Thesis - Leiden University, Faculty of Science

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08 November 2016

Charting Biologically Relevant Spirocyclic Compound Space

G. Müller, T. Berkenbosch, J. Benningshof, D. Stumpfe, J. Bajorath 
Chemistry
doi: 10.1002/chem.201604714 2016 November 8 (epub ahead of print)

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02 November 2016

Easy Synthesis of Two Positional Isomeric Tetrazole Libraries

Yuanze Wang, Pravin Patil, Alexander Dömling
Synthesis 2016;48(21):3701-3712
doi: https://doi.org/10.1055/s-0035-1562435 2016 November 2

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20 October 2016

Ugi-Type Reactions of Spirocyclic Indolenines as a Platform for Compound Library Generation

Verónica Estévez, Laura Kloeters, Natalia Kwietniewska, Esther Vicente-García, Eelco Ruijter, Romano V.A. Orru
Synlett 2017;28(03):376-380
doi: https://doi.org/10.1055%2Fs-0036-1588084 2016 October 20

 

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05 October 2016

The SULSA Assay Development Fund: accelerating translation of new biology from academia to pharma

S.P. McElroy, P.S. Jones, D.V. Barrault
Drug Discov Today. 2016 Oct 5
doi:10.1016/j.drudis.2016.09.028 Epub 2016 October 5

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09 September 2016

Cleavable β-Cyanoethyl Isocyanide in the Ugi Tetrazole Reaction

E. Kroon, K. Kurpiewska, J. Kalinowska-Tłuścik and A. Dömling 
Org. Lett., Article ASAP
doi: 10.1021/acs.orglett.6b01826 2016 September 9

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06 September 2016

Artificial Macrocycles by Ugi Reaction and Passerini Ring Closure

E.M.M. Abdelraheem, K. Kurpiewska, J. Kalinowska-Tłuścik and A. Dömling 
J Org Chem. 2016 Sep 15 
doi:10.1021/acs.joc.6b01430 Epub 2016 September 6

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01 September 2016

Public–private partnerships in lead discovery: overview and case studies

Matthias Gottwald, Andreas Becker, Inke Bahr, Anke Mueller‐Fahrnow
Archiv der Pharmazie 2016;349(9):692-697
doi: https://doi.org/10.1002/ardp.201600078 2016 September 1

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