Publications

This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication. 

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08 November 2016

Charting Biologically Relevant Spirocyclic Compound Space

G. Müller, T. Berkenbosch, J. Benningshof, D. Stumpfe, J. Bajorath 
Chemistry
doi: 10.1002/chem.201604714 2016 November 8 (epub ahead of print)

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02 November 2016

Easy Synthesis of Two Positional Isomeric Tetrazole Libraries

Yuanze Wang, Pravin Patil, Alexander Dömling
Synthesis 2016;48(21):3701-3712
doi: https://doi.org/10.1055/s-0035-1562435 2016 November 2

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20 October 2016

Ugi-Type Reactions of Spirocyclic Indolenines as a Platform for Compound Library Generation

Verónica Estévez, Laura Kloeters, Natalia Kwietniewska, Esther Vicente-García, Eelco Ruijter, Romano V.A. Orru
Synlett 2017;28(03):376-380
doi: https://doi.org/10.1055%2Fs-0036-1588084 2016 October 20

 

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05 October 2016

The SULSA Assay Development Fund: accelerating translation of new biology from academia to pharma

S.P. McElroy, P.S. Jones, D.V. Barrault
Drug Discov Today. 2016 Oct 5
doi:10.1016/j.drudis.2016.09.028 Epub 2016 October 5

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09 September 2016

Cleavable β-Cyanoethyl Isocyanide in the Ugi Tetrazole Reaction

E. Kroon, K. Kurpiewska, J. Kalinowska-Tłuścik and A. Dömling 
Org. Lett., Article ASAP
doi: 10.1021/acs.orglett.6b01826 2016 September 9

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06 September 2016

Artificial Macrocycles by Ugi Reaction and Passerini Ring Closure

E.M.M. Abdelraheem, K. Kurpiewska, J. Kalinowska-Tłuścik and A. Dömling 
J Org Chem. 2016 Sep 15 
doi:10.1021/acs.joc.6b01430 Epub 2016 September 6

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01 September 2016

Public–private partnerships in lead discovery: overview and case studies

Matthias Gottwald, Andreas Becker, Inke Bahr, Anke Mueller‐Fahrnow
Archiv der Pharmazie 2016;349(9):692-697
doi: https://doi.org/10.1002/ardp.201600078 2016 September 1

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27 August 2016

Expedient synthesis of an atypical oxazolidinone compound library

S.J. Cully, T.E. Storra, M.J. Rawling, I.R. Abeysen, D. Hamza, G. Jones, C.A. Pearce, A. Quddus, W. Lewis and R.A. Stockman
Bioorg Med Chem. 2016 Aug 27
doi: 10.1039/c6cc04662b 2016 August 27

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18 July 2016

A biosynthesis-inspired approach to over twenty diverse natural product-like scaffolds

J.D. Firth, P.G.E. Craven, M. Lilburn, A.Pahl, S. P. Marsden and A. Nelson
Chem. Commun., 2016, 52, 9837
doi:10.1039/c6cc04662b Epub 2016 July 18

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24 June 2016

A metal-catalyzed enyne-cyclization step for the synthesis of bi- and tricyclic scaffolds amenable to molecular library production

P. Wu, M.Å. Petersen, A.E. Cohrt, R. Petersen, R. Morgentin, H. Lemoine, C. Roche, A. Willaume, M.H. Clausen and T.E. Nielsen 
Org. Biomol. Chem., 2016,14, 6947-6950 
doi: 10.1039/C6OB01148A 2016 June 24

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