This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication.
Densely functionalised spirocyclic oxetane-piperidine scaffolds for drug discovery
Gemma C. Geary, Andrew Nortcliffe, Christopher A. Pearce, Daniel Hamza, Geraint Jones, Christopher J. Moody
Bioorganic & Medicinal Chemistry 2018;26(4):791-797
doi: https://doi.org/10.1016/j.bmc.2017.12.012 2018 February 15
Two-Step Macrocycle Synthesis by Classical Ugi Reaction
Eman M. M. Abdelraheem, Samad Khaksar, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Shabnam Shaabani, Alexander Dömling
Journal of Organic Chemistry 2018;83(3):1441–1447
doi: 10.1021/acs.joc.7b02984 2018 January 12
Concise synthesis of macrocycles by multicomponent reactions
Eman M. M. Abdelraheem, Samad Khaksar, Alexander Dömling
Synthesis 2018;50(5):1027-1038
doi: 10.1055/s-0036-1590946 2018 January 10
Library-to-Library Synthesis of Highly Substituted α-Aminomethyl Tetrazoles via Ugi Reaction
Pravin Patil, Bhupendra Mishra, Gitanjali Sheombarsing, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Alexander Dömling
ACS Combinatorial Science 2018;20(2):70–74
doi: 10.1021/acscombsci.7b00137 2017 December 7
Microwave-assisted Diastereoselective Two-step Three-component Synthesis for Rapid Access to Drug-like Libraries of Substituted 3-Amino-β-lactams
Ugi Multicomponent Reaction Based Synthesis of Medium-Sized Rings
Eman M. M. Abdelraheem, Rudrakshula Madhavachary, Arianna Rossetti, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Shabnam Shaabani, Alexander Dömling
Organic Letters 2017;19(22):6176–6179
doi: 10.1021/acs.orglett.7b03094 2017 October 30
Diastereoselective One Pot Five-Component Reaction toward 4-(Tetrazole)-1,3-Oxazinanes
Ajay L. Chandgude, Daniele Narducci, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścikb, Alexander Dömling
RSC Advances 2017;79:49995-49998
doi: 10.1039/C7RA07392E 2017 October 26, Open Access
Synthesis and Demonstration of the Biological Relevance of sp3-rich Scaffolds Distantly Related to Natural Product Frameworks
Daniel J. Foley, Philip G. E. Craven, Patrick M. Collins, Richard G. Doveston, Anthony Aimon, Romain Talon, Ian Churcher, Frank von Delft, Stephen P. Marsden, Adam Nelson
Chem. Eur. J. 2017;23,15227
doi: https://doi.org/10.1002/chem.201704169 2017 October 10, Open Access
Privileged heterocycles: bioactivity and synthesis of 1,9-diazaspiro 5.5 undecane-containing compounds
Daniel Blanco-Ania, Rik Heus, Floris P.J.T. Rutjes
Chemistry of Heterocyclic Compounds 2017;53(8):827–845
doi: https://doi.org/10.1007/s1059 2017 October 5
Piperidine and octahydropyrano[3,4-c]pyridine scaffolds for drug-like molecular libraries of the European Lead Factory
B.D. Narhe, A.C. Breman, J. Padwal, D.A.L. Vandenput, J.M. Scheidt, J.C.J. Benningshof, G.A. van der Marel, H.S. Overkleeft, M. van der Stelt, D.V. Filippov
Bioorganic & Medicinal Chemistry 2017; 25:5160–5170
doi: 10.1016/j.bmc.2017.07.016 2017 October 1
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