This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication.
Design and synthesis of a fragment set based on twisted bicyclic lactams
H. Hassan, S.P. Marsden, A. Nelson
Bioorganic & Medicinal Chemistry 2018;26(11):3030-3033
doi: 10.1016/j.bmc.2018.02.027 2018 February 22
Using Microscale Thermophoresis to Characterize Hits from High-Throughput Screening: A European Lead Factory Perspective
Synthesis of Highly Substituted Imidazole Uracil Containing Molecules via Ugi-4CR and Passerini-3CR
Rudrakshula Madhavachary, Tryfon Zarganes-Tzitzikas, Pravin Patil, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Alexander Dömling
ACS Combinatorial Science 2018;20(4):192–196
doi: 10.1021/acscombsci.7b00145 2018 February 19
Densely functionalised spirocyclic oxetane-piperidine scaffolds for drug discovery
Gemma C. Geary, Andrew Nortcliffe, Christopher A. Pearce, Daniel Hamza, Geraint Jones, Christopher J. Moody
Bioorganic & Medicinal Chemistry 2018;26(4):791-797
doi: https://doi.org/10.1016/j.bmc.2017.12.012 2018 February 15
Two-Step Macrocycle Synthesis by Classical Ugi Reaction
Eman M. M. Abdelraheem, Samad Khaksar, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Shabnam Shaabani, Alexander Dömling
Journal of Organic Chemistry 2018;83(3):1441–1447
doi: 10.1021/acs.joc.7b02984 2018 January 12
Concise synthesis of macrocycles by multicomponent reactions
Eman M. M. Abdelraheem, Samad Khaksar, Alexander Dömling
Synthesis 2018;50(5):1027-1038
doi: 10.1055/s-0036-1590946 2018 January 10
Library-to-Library Synthesis of Highly Substituted α-Aminomethyl Tetrazoles via Ugi Reaction
Pravin Patil, Bhupendra Mishra, Gitanjali Sheombarsing, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Alexander Dömling
ACS Combinatorial Science 2018;20(2):70–74
doi: 10.1021/acscombsci.7b00137 2017 December 7
Microwave-assisted Diastereoselective Two-step Three-component Synthesis for Rapid Access to Drug-like Libraries of Substituted 3-Amino-β-lactams
Ugi Multicomponent Reaction Based Synthesis of Medium-Sized Rings
Eman M. M. Abdelraheem, Rudrakshula Madhavachary, Arianna Rossetti, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścik, Shabnam Shaabani, Alexander Dömling
Organic Letters 2017;19(22):6176–6179
doi: 10.1021/acs.orglett.7b03094 2017 October 30
Diastereoselective One Pot Five-Component Reaction toward 4-(Tetrazole)-1,3-Oxazinanes
Ajay L. Chandgude, Daniele Narducci, Katarzyna Kurpiewska, Justyna Kalinowska-Tłuścikb, Alexander Dömling
RSC Advances 2017;79:49995-49998
doi: 10.1039/C7RA07392E 2017 October 26, Open Access
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