This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication. 
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06 October 2017

Synthesis and Demonstration of the Biological Relevance of sp3-rich Scaffolds Distantly Related to Natural Product Frameworks

Daniel J. Foley, Philip G. E. Craven, Patrick M. Collins, Richard G. Doveston, Anthony Aimon, Romain Talon, Ian Churcher, Frank von Delft, Stephen P. Marsden, Adam Nelson
Chem. Eur. J. 2017;23,15227
doi: 2017 October 10, Open Access

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05 October 2017

Privileged heterocycles: bioactivity and synthesis of 1,9-diazaspiro 5.5 undecane-containing compounds

Daniel Blanco-Ania, Rik Heus, Floris P.J.T. Rutjes
Chemistry of Heterocyclic Compounds 2017;53(8):827–845
doi: 2017 October 5

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01 October 2017

Piperidine and octahydropyrano[3,4-c]pyridine scaffolds for drug-like molecular libraries of the European Lead Factory

B.D. Narhe, A.C. Breman, J. Padwal, D.A.L. Vandenput, J.M. Scheidt, J.C.J. Benningshof, G.A. van der Marel, H.S. Overkleeft, M. van der Stelt, D.V. Filippov
Bioorganic & Medicinal Chemistry 2017; 25:5160–5170
doi: 10.1016/j.bmc.2017.07.016 2017 October 1

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05 September 2017

C−H Insertion as a Key Step to Spiro-Oxetanes, Scaffolds for Drug Discovery

Simon M. Nicolle, Andrew Nortcliffe, Hannah E. Bartrum, William Lewis, Christopher J. Hayes, Christopher J. Moody
Chem. Eur. J. 2017;23,13623
doi: 2017 September 5

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01 August 2017

Two-Step Synthesis of Complex Artificial Macrocyclic Compounds

Rudrakshula Madhavachary, Eman M. M. Abdelraheem, Arianna Rossetti, Aleksandra Twarda‐Clapa, Bogdan Musielak, Katarzyna Kurpiewska, Justyna Kalinowska‐Tłuścik, Tad A. Holak, Alexander Dömling  
Angew Chem Int Ed Engl 2017;56(36):10725-10729
doi: 2017 August 1

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12 July 2017

With unprotected amino acids to tetrazolo peptidomimetics

Rudrakshula Madhavachary, Qian Wanga, Alexander Dömling
Chemical Communications 2017;53:8549-8552 
doi: 10.1039/C7CC03370B 2017 July 12

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29 June 2017

Diastereoselective synthesis of novel heterocyclic scaffolds through tandem Petasis 3-component/intramolecular Diels–Alder and ROM–RCM reactions

Mette Ishoey, Rico G. Petersen,  Michael Å. Petersen, Peng Wu,  Mads H. Clausen, Thomas E. Nielsen
Chemical Communications 2017;53:9410-9413 
doi: 10.1039/C7CC02948A 2017 June 29  

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13 June 2017

Reference Module in Chemistry, Molecular Sciences and Chemical Engineering

F. Giordanetto, P. Jones, A. Nelson, J. Benningshof, G. Müller, A. Pannifer and D.Tzalis
Comprehensive Medicinal Chemistry III 2017, 505-519
doi:10.1016/B978-0-12-409547-2.12303-0 2017 June 13

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05 June 2017

Sulfur-Switch Ugi-Reaction For Macrocyclic Disulfide-Bridged Peptidomimetics

T. M. Vishwanatha, E. Bergamaschi and A. Dömling
Organic Letters Article ASAP 2017
doi: 10.1021/acs.orglett.7b01324 2017 June 5

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18 May 2017

Highly Stereoselective Synthesis of a Compound Collection Based on the Bicyclic Scaffolds of Natural Products

M. Annamalai, S. Hristeva, M. Bielska, R. Ortega and K. Kumar
Molecules 2017, 22, 827
doi: 10.3390/molecules22050827 2017 May 18