Publications

This is a non exhaustive list of publications related to ELF work published in scientific journals. Please contact the programme office if you miss a relevant publication. 
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27 February 2017

Ammonia-Promoted One-Pot Tetrazolopiperidinone Synthesis by Ugi Reaction

P. Patil, K. Kurpiewska, J. Kalinowska-Tłusćik and A. Dömling
ACS Comb. Sci. 2017, 19, 343−350
doi: 10.1021/acscombsci.7b00033 2017 February 27

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24 February 2017

Synthesis of 4-aminotetrahydropyran scaffolds for drug discovery

A. Nortcliffe, G.D.S. Milne, D. Hamza and C.J. Moody 
Bioorganic & Medicinal Chemistry 25 (2017) 2218–2225
doi: 10.1016/j.bmc.2017.02.039 2017 February 24

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09 February 2017

Two Cycles with One Catch: Hydrazine in Ugi 4-CR and Its Postcyclizations

Y. Wang, P. Patil, K. Kurpiewska, J. Kalinowska-Tluscik and A. Dömling
ACS Comb Sci. 2017 Mar 13;19(3):193-198
doi: 10.1021/acscombsci.7b00009 2017 February 9

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09 February 2017

Cysteine Isocyanide in Multicomponent Reaction: Synthesis of Peptido-Mimetic 1,3-Azoles

T.M. Vishwanatha, A. Domling, K. Kurpiewska, J. Kalinowska-Tluscik
J Org Chem. 2017;82(18):9585-9594
doi: 10.1021/acs.joc.7b01615 2017 September 15

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19 January 2017

The European Lead Factory: A Blueprint for Public–Private Partnerships in Early Drug Discovery

A. Karawajczyk, K.M. Orrling, J.B.S. de Vlieger, T. Rijnders and D. Tzalis
Front. Med. 2017 3 (75)
doi: 10.3389/fmed.2016.00075 2017 January 19

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19 January 2017

De Novo Assembly of Highly Substituted Morpholines and Piperazines

P. Patil, R. Madhavachary, K. Kurpiewska, J. Kalinowska-Tłuścik and A. Dömling
Org Lett
doi: 10.1021/acs.orglett.6b03807 2017 January 19

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18 January 2017

An Enantio- and Diastereoselective Mannich/Pictet-Spengler Sequence To Form Spiro piperidine-pyridoindoles and Application to Library Synthesis

Alejandra Riesco‐Domínguez, Nick van der Zwaluw, Daniel Blanco‐Ania, Floris P. J. T. Rutjes
European Journal of Organic Chemistry 2017;3:662-670
doi: https://doi.org/10.1002/ejoc.201601508 2017 January 18

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19 December 2016

Synthesis of Epibatidine Analogues by Pyrrole Diels–Alder Reactions: Rapid Access to Azabicyclo[2.2.1]heptane and 3,8-Diazabicyclo[3.2.1]octane Scaffolds for Library Synthesis

A.T. Murray, E. Packard, A. Nortcliffe, W. Lewis, D. Hamza, G. Jones, C.J. Moody
Eur. J. Org. Chem. 2017, 138–148
doi: 10.1002/ejoc.201601177 2016 December 19

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01 December 2016

Unconventional Passerini Reaction toward α‑Aminoxy-amides

A.L. Chandgude and A.S.S. Dömling
Org. Lett., 2016, 18 (24), pp 6396–6399
doi: 10.1021/acs.orglett.6b03293 2016 December 1

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01 December 2016

Discovery of novel inhibitors to investigate diacylglycerol lipases and α/β hydrolase domain 16A

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